Highly efficient methods for the one-pot synthesis of beta-substituted enones.

نویسندگان

  • William J Kerr
  • Colin M Pearson
  • Graeme J Thurston
چکیده

A mild and practically-convenient one-pot procedure for the direct beta-substitution of enones has been developed using a conjugate addition-oxidation strategy with a full range of copper-based reagents and N-tert-butylphenylsulfinimidoyl chloride; alkyl- and aryl-substituted enones are delivered in good to excellent yields.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 4 1  شماره 

صفحات  -

تاریخ انتشار 2006